Timapiprant Sodium

Catalogue Number: E0809-SEL

Manufacturer:Selleck Chemicals
Shelf Life:36 months
Molecular Formula:C21H17FN2O2.Na
Type:Other Proteins
Alias:OC000459 sodium
Shipping Condition:Blue Ice
Unit(s): 5 mg

Additional Text

CAS Number

950688-14-9

Short Description

Timapiprant sodium (OC000459 sodium), a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist, potently displaces [3H]PGD2 from human recombinant DP2, rat recombinant DP2, and human native DP2 with Ki values of 13, 3 and 4 nM, respectively.

Smile String

[NaH].CC1=C(CC2=NC3=C(C=CC=C3)C=C2)C4=CC(=CC=C4[N]1CC(O)=O)F

Storage Note

3 years -20°C powder