Rolapitant
Catalogue Number: S5476-SEL
| Manufacturer: | Selleck Chemicals |
| Shelf Life: | 36 months |
| Molecular Formula: | C25H26F6N2O2 |
| Type: | Other Inhibitors |
| Alias: | SCH-619734 |
| Shipping Condition: | Blue Ice |
| Unit(s): | 5 mg, 1 g, 100 mg |
Additional Text
Short Description
Rolapitant (SCH-619734) is a selective and competitive antagonist of human substance P/NK1 receptors with antiemetic activity. It has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold, as well as preferential affinity for human, guinea pig, gerbil and monkey NK1 receptors over rat, mouse and rabbit.
Smile String
CC(C1=CC(=CC(=C1)C(F)(F)F)C(F)(F)F)OCC2(CCC3(CCC(=O)N3)CN2)C4=CC=CC=C4
Storage Note
3 years -20°C powder
Inhibitor Handling Instructions
SUPPORT
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PRODUCT
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DELIVERY
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