Catalogue Number: S8409-SEL
| Manufacturer: | Selleck Chemicals |
| Shelf Life: | 36 months |
| Molecular Formula: | C17H13ClNO5P |
| Type: | Other Inhibitors |
| Alias: | 2-naphthol-AS-E-phosphate |
| Shipping Condition: | Blue Ice |
| Unit(s): | 10 mg, 10 mM/1 ml |
KG-501 is a cAMP response element-binding protein (CREB) inhibitor that disrupts CREB-dependent transcription (Ki = 10 µM) and CREB:CBP interaction (Ki = 50 µM). It also disrupts phospho (Ser-133) CREB binding to KIX with a Ki of ~90 µM, using concentrations of CREB that were within the linear range of the binding assay.
C1=CC=C2C=C(C(=CC2=C1)C(=O)NC3=CC=C(C=C3)Cl)OP(=O)(O)O
3 years -20°C powder