Tanzisertib(CC-930)
Catalogue Number: S8490-SEL
| Manufacturer: | Selleck Chemicals |
| Type: | Biochemicals |
| Shipping Condition: | Blue Ice |
| Unit(s): | 5 mg, 25 mg, 10 mM/1 ml |
Description
Description: Tanzisertib (CC-930, JNK-930, JNKI-1) is kinetically competitive with ATP in the JNK-dependent phosphorylation of the protein substrate c-Jun and potent against all isoforms of JNK (Ki(JNK1) = 44 +/- 3 nM, IC50(JNK1) = 61 nM, Ki(JNK2) = 6.2 +/- 0.6 nM, IC50(JNK2) = 5 nM, IC50(JNK3) = 5 nM) and selective against MAP kinases ERK1 and p38a with IC50 of 0.48 and 3.4 µM respectively.
S8490 MSDS
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